8- (3-Chlorostyryl) caffeine [CAS 148589-13-3]
8- (3-Chlorostyryl) caffeine [CAS 148589-13-3]
SKU:QM-0083071
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Product Details
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Description
8- (3-Chlorostyryl) caffeine (CSC) is an adenosine antagonist with selective activity at the A2a adenosine receptor. 8- (3-Chlorostyryl) caffeine showed 520-fold selectivity in radioligand binding experiments in rat brain. Antagonism of adenylylase by 8- (3-Chlorostyryl) caffeine shows 22-fold selectivity in rat chromaffin cells When 8- (3-Chlorostyryl) caffeine is co-administered with the A1-selective antagonist CPX, It can also further increase exercise activity. 8- (3-Chlorostyryl) caffeine exhibits good MAO-B inhibitory activity in primate mitochondria. 8- (3-Chlorostyryl) caffeine also has excellent A2A receptor affinity[1].
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CAS Number
[148589-13-3]
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Molecular Formula
C16H15ClN4O2
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Molecular Weight
330.77
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Smiles
O=C(N(C1=C(C2=O)N(C(/C=C/C3=CC=CC(Cl)=C3)=N1)C)C)N2C
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Target
Endogenous Metabolite
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Shipping Conditions
Room temperature
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8- (3-Chlorostyryl) caffeine [CAS 148589-13-3]
8- (3-Chlorostyryl) caffeine is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.