Collection: Bioactive Small Molecules
Explore QuantiMol's extensive range of bioactive small molecules for life science research, pathway studies, high-throughput screening, and drug discovery applications. This collection spans the full spectrum of pharmacological activity — including enzyme inhibitors, kinase inhibitors, protease inhibitors, receptor agonists and antagonists, ion channel modulators, epigenetic probes, and signalling pathway tool compounds — covering virtually every major biological target class relevant to modern biomedical research.
Each bioactive small molecule supplied by QuantiMol is rigorously characterised for purity, identity, and biological activity, giving researchers the confidence to use them as primary pharmacological tools in mechanistic studies, target validation, and lead optimisation workflows. Whether you are dissecting a signalling cascade, profiling off-target effects, or building a focused screening library, QuantiMol's bioactive small molecules provide the chemical precision your research demands.
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β-catenin inhibitory peptoid [CAS 2579070-02-1]
CAS: 2579070-02-1 | SKU: QM-0025230 | Size: 1 Each Price on request -
α-Synuclein inhibitor 14 [CAS 408324-13-0]
CAS: 408324-13-0 | SKU: QM-0023369 | Size: 1 Each Price on request -
β2AR agonist 5 [CAS 2759727-47-2]
CAS: 2759727-47-2 | SKU: QM-0015918 | Size: 1 Each Price on request -
α2AR agonist 2 [CAS 719277-27-7]
CAS: 719277-27-7 | SKU: QM-0015098 | Size: 1 Each Price on request -
α-Synuclein inhibitor 15 [CAS 414880-30-1]
CAS: 414880-30-1 | SKU: QM-0013035 | Size: 1 Each Price on request -
αMβ2 integrin agonist-1
SKU: QM-0013016 | Size: 1 Each Price on request -
α5β1 integrin agonist-2
SKU: QM-0013015-01 | Size: 5 mg£476.46 GBP -
α4β1 antagonist-1
SKU: QM-0013014 | Size: 1 Each Price on request -
YTHDF2 ligand-1 [CAS 3093182-34-1]
CAS: 3093182-34-1 | SKU: QM-0012730-01 | Size: 5 mg£370.76 GBP -
α5-GABAA receptor modulator 1
SKU: QM-0009574 | Size: 1 Each Price on request -
α-syn aggregation inhibitor-1
SKU: QM-0009265 | Size: 1 Each Price on request -
β-Catenin modulator-8 [CAS 902586-39-4]
CAS: 902586-39-4 | SKU: QM-0008903 | Size: 1 Each Price on request -
β-Secretase Inhibitor IV (Standard) [CAS 797035-11-1]
CAS: 797035-11-1 | SKU: QM-0002305 | Size: 1 Each Price on request -
γ-Secretase modulator 4 [CAS 1420200-82-3]
CAS: 1420200-82-3 | SKU: QM-0142451-01 | Size: 1 mg£577.31 GBP -
σ1 Receptor antagonist-1 [CAS 1204401-49-9]
CAS: 1204401-49-9 | SKU: QM-0112884-01 | Size: 5 mg£146.50 GBP -
α7 Nicotinic receptor agonist-1 [CAS 220100-05-0]
CAS: 220100-05-0 | SKU: QM-0149648-01 | Size: 5 mg£452.17 GBP -
β-FXR antagonist 1 [CAS 2295804-92-9]
CAS: 2295804-92-9 | SKU: QM-0150540-01 | Size: 5 mg£539.64 GBP -
α-Synuclein inhibitor 11
SKU: QM-0153508-01 | Size: 5 mg£263.84 GBP -
YAP/TAZ inhibitor-3 [CAS 2506273-81-8]
CAS: 2506273-81-8 | SKU: QM-0156055-01 | Size: 5 mg£414.50 GBP -
α-Synuclein inhibitor 10 [CAS 3050715-65-3]
CAS: 3050715-65-3 | SKU: QM-0152258-01 | Size: 5 mg£301.50 GBP -
α5β1 integrin agonist-1 [CAS 2756557-83-0]
CAS: 2756557-83-0 | SKU: QM-0146845-01 | Size: 1 mg£476.46 GBP -
α7 nAchR-JAK2-STAT3 agonist 1 [CAS 2108714-20-9]
CAS: 2108714-20-9 | SKU: QM-0075255-01 | Size: 5 mg£652.64 GBP -
δ-Secretase inhibitor 11 [CAS 842964-18-5]
CAS: 842964-18-5 | SKU: QM-0141339-01 | Size: 10 mg£89.13 GBP -
α2β1 Integrin Ligand Peptide (TFA)
SKU: QM-0196447-01 | Size: 1 mg£78.82 GBP -
β-Secretase Inhibitor IV [CAS 797035-11-1]
CAS: 797035-11-1 | SKU: QM-0081148-01 | Size: 1 mg£351.32 GBP -
β-Catenin modulator-2 [CAS 1015858-71-5]
CAS: 1015858-71-5 | SKU: QM-0151249-01 | Size: 5 mg£401.13 GBP -
α7β1 integrin modulator-1 [CAS 849121-82-0]
CAS: 849121-82-0 | SKU: QM-0156358-01 | Size: 5 mg£78.82 GBP -
ZL-12A probe
SKU: QM-0161283-01 | Size: 1 mg£1,656.23 GBP -
β-Secretase Inhibitor III [CAS 2760674-85-7]
CAS: 2760674-85-7 | SKU: QM-0063806 | Size: 1 Each Price on request -
γ-Secretase modulator 16 [CAS 884599-96-6]
CAS: 884599-96-6 | SKU: QM-0136960 | Size: 1 Each Price on request -
α2AR agonist 1
SKU: QM-0153235 | Size: 1 Each Price on request -
α-Synuclein modulator 1 [CAS 3058709-40-0]
CAS: 3058709-40-0 | SKU: QM-0133147 | Size: 1 Each Price on request -
β2AR ligand 1 [CAS 3051498-44-0]
CAS: 3051498-44-0 | SKU: QM-0132111 | Size: 1 Each Price on request -
α-Synuclein inhibitor 4 [CAS 2489813-08-1]
CAS: 2489813-08-1 | SKU: QM-0067471 | Size: 1 Each Price on request -
σ1 Receptor/μ Opioid receptor modulator 2 [CAS 3009018-61-2]
CAS: 3009018-61-2 | SKU: QM-0073595 | Size: 1 Each Price on request -
μ opioid receptor agonist 2 [CAS 2671755-38-5]
CAS: 2671755-38-5 | SKU: QM-0065092 | Size: 1 Each Price on request -
YAP/TAZ inhibitor-4
SKU: QM-0126181 | Size: 1 Each Price on request -
β-Catenin modulator-3 [CAS 1015858-17-9]
CAS: 1015858-17-9 | SKU: QM-0070727 | Size: 1 Each Price on request -
δ opioid receptor antagonist 1
SKU: QM-0122210 | Size: 1 Each Price on request -
α-Synuclein inhibitor 13
SKU: QM-0121938 | Size: 1 Each Price on request -
[Tyr0] Gastric Inhibitory Peptide (23-42), human [CAS 121765-67-1]
CAS: 121765-67-1 | SKU: QM-0076383 | Size: 1 Each Price on request -
α4 integrin receptor antagonist 3 [CAS 863226-74-8]
CAS: 863226-74-8 | SKU: QM-0120647 | Size: 1 Each Price on request -
σ1 Receptor antagonist 4 [CAS 362512-81-0]
CAS: 362512-81-0 | SKU: QM-0119784 | Size: 1 Each Price on request -
γ-Secretase modulator 11 [CAS 2434630-29-0]
CAS: 2434630-29-0 | SKU: QM-0067513 | Size: 1 Each Price on request -
μ opioid receptor agonist 1 [CAS 2667632-83-7]
CAS: 2667632-83-7 | SKU: QM-0065091 | Size: 1 Each Price on request -
β-Catenin modulator-5 [CAS 902168-07-4]
CAS: 902168-07-4 | SKU: QM-0070729 | Size: 1 Each Price on request -
β2AR/M3-receptor agonist-1 [CAS 1206887-00-4]
CAS: 1206887-00-4 | SKU: QM-0067954 | Size: 1 Each Price on request -
α1B-AR antagonist 1 [CAS 874129-03-0]
CAS: 874129-03-0 | SKU: QM-0114441 | Size: 1 Each Price on request -
γ-Secretase modulator 14 [CAS 1420200-85-6]
CAS: 1420200-85-6 | SKU: QM-0067872 | Size: 1 Each Price on request -
α-Synuclein inhibitor 3 [CAS 2687831-18-9]
CAS: 2687831-18-9 | SKU: QM-0067457 | Size: 1 Each Price on request -
β2AR antagonist 1 [CAS 2135743-21-2]
CAS: 2135743-21-2 | SKU: QM-0109152 | Size: 1 Each Price on request -
β-Secretase inhibitor [CAS 350228-37-4]
CAS: 350228-37-4 | SKU: QM-0109125-01 | Size: 1 mg£232.25 GBP -
γ-Secretase modulator 12 [CAS 2204249-82-9]
CAS: 2204249-82-9 | SKU: QM-0066640 | Size: 1 Each Price on request -
γ-Secretase modulator 11 (hydrochloride) [CAS 2434630-30-3]
CAS: 2434630-30-3 | SKU: QM-0067514 | Size: 1 Each Price on request -
β-Catenin modulator-7 [CAS 2892294-93-6]
CAS: 2892294-93-6 | SKU: QM-0103211 | Size: 1 Each Price on request -
α-Synuclein inhibitor 6 [CAS 2489813-02-5]
CAS: 2489813-02-5 | SKU: QM-0067473 | Size: 1 Each Price on request -
β2AR agonist /M-receptor antagonist-1 [CAS 2772700-36-2]
CAS: 2772700-36-2 | SKU: QM-0067956 | Size: 1 Each Price on request -
αvβ6 integrin inhibitor 2 [CAS 313709-47-6]
CAS: 313709-47-6 | SKU: QM-0070781 | Size: 1 Each Price on request -
β-Secretase Inhibitor II [CAS 263563-09-3]
CAS: 263563-09-3 | SKU: QM-0063091 | Size: 1 Each Price on request -
γ-Secretase modulator 13 [CAS 1353570-40-7]
CAS: 1353570-40-7 | SKU: QM-0068779-01 | Size: 1 mg£734.04 GBP -
α-Synuclein inhibitor 7 [CAS 2489813-04-7]
CAS: 2489813-04-7 | SKU: QM-0067474 | Size: 1 Each Price on request -
σ1 Receptor/μ Opioid receptor modulator 1 [CAS 2412700-00-4]
CAS: 2412700-00-4 | SKU: QM-0067387 | Size: 1 Each Price on request -
α-Synuclein inhibitor 5 [CAS 2489813-11-6]
CAS: 2489813-11-6 | SKU: QM-0067472 | Size: 1 Each Price on request -
μ opioid receptor agonist 3 [CAS 2378397-91-0]
CAS: 2378397-91-0 | SKU: QM-0071711 | Size: 1 Each Price on request -
β2AR agonist 4
SKU: QM-0098552 | Size: 1 Each Price on request -
α2β1 Integrin Ligand Peptide [CAS 134580-64-6]
CAS: 134580-64-6 | SKU: QM-0001292-01 | Size: 1 mg£78.82 GBP -
α2δ ligand 1 [CAS 313653-15-5]
CAS: 313653-15-5 | SKU: QM-0096789 | Size: 1 Each Price on request -
β-AR antagonist 2 [CAS 2779507-62-7]
CAS: 2779507-62-7 | SKU: QM-0096263 | Size: 1 Each Price on request -
β2AR agonist 2
SKU: QM-0068560 | Size: 1 Each Price on request -
β-catenin modulator IIa-661 [CAS 1015859-04-7]
CAS: 1015859-04-7 | SKU: QM-0075637-01 | Size: 1 mg£92.50 GBP -
β2AR agonist 3 [CAS 2304455-74-9]
CAS: 2304455-74-9 | SKU: QM-0068561 | Size: 1 Each Price on request -
β3-AR agonist 3 [CAS 883724-08-1]
CAS: 883724-08-1 | SKU: QM-0058294 | Size: 1 Each Price on request -
β3-AR agonist 2 [CAS 340757-05-3]
CAS: 340757-05-3 | SKU: QM-0091562 | Size: 1 Each Price on request -
β-Catenin modulator-1 [CAS 1053086-89-7]
CAS: 1053086-89-7 | SKU: QM-0070726 | Size: 1 Each Price on request -
α7 nAChR Modulator-2
SKU: QM-0090633 | Size: 1 Each Price on request -
α7 nAChR Modulator-3
SKU: QM-0090067 | Size: 1 Each Price on request -
α-Synuclein inhibitor 8 [CAS 2883627-64-1]
CAS: 2883627-64-1 | SKU: QM-0070145 | Size: 1 Each Price on request -
β-Catenin modulator-4 [CAS 901751-85-7]
CAS: 901751-85-7 | SKU: QM-0070728 | Size: 1 Each Price on request -
ZBP1/RIP3/MLKL activator 1
SKU: QM-0089589-01 | Size: 5 mg£238.32 GBP -
β-Glucocerebrosidase modulator 1 [CAS 3080715-77-8]
CAS: 3080715-77-8 | SKU: QM-0089097-01 | Size: 5 mg£1,719.41 GBP -
α2C adrenoceptor agonist 1 [CAS 928115-79-1]
CAS: 928115-79-1 | SKU: QM-0088530 | Size: 1 Each Price on request -
γ-Secretase modulator 10 [CAS 2694817-84-8]
CAS: 2694817-84-8 | SKU: QM-0066217 | Size: 1 Each Price on request -
α2A-AR agonist 1 [CAS 2971825-58-6]
CAS: 2971825-58-6 | SKU: QM-0087261-01 | Size: 5 mg£238.32 GBP -
β3-AR agonist 1 [CAS 1283125-73-4]
CAS: 1283125-73-4 | SKU: QM-0057108 | Size: 1 Each Price on request -
β-Secretase Inhibitor I [CAS 1818239-19-8]
CAS: 1818239-19-8 | SKU: QM-0060873 | Size: 1 Each Price on request -
α-Synuclein inhibitor 9 [CAS 1510825-03-2]
CAS: 1510825-03-2 | SKU: QM-0068414 | Size: 1 Each Price on request -
β2AR/M-receptor agonist-1 [CAS 2230520-62-2]
CAS: 2230520-62-2 | SKU: QM-0067952 | Size: 1 Each Price on request -
α-Synuclein inhibitor 12
SKU: QM-0080099 | Size: 1 Each Price on request -
σ1 Receptor ligand 1
SKU: QM-0078552 | Size: 1 Each Price on request -
Vipivotide tetraxetan Ligand-Linker Conjugate [CAS 1703768-74-4]
CAS: 1703768-74-4 | SKU: QM-0017305-01 | Size: 5 mg£282.06 GBP -
VDR ligand-1
SKU: QM-0016015 | Size: 1 Each Price on request -
WDR5 probe 1
SKU: QM-0015746 | Size: 1 Each Price on request -
V1b Receptor antagonist-1 [CAS 1056550-56-1]
CAS: 1056550-56-1 | SKU: QM-0015336 | Size: 1 Each Price on request -
VDR agonist 4
SKU: QM-0015150 | Size: 1 Each Price on request -
WRN inhibitor 19
SKU: QM-0014071 | Size: 1 Each Price on request -
URAT1 inhibitor 13 [CAS 2816864-54-5]
CAS: 2816864-54-5 | SKU: QM-0013637 | Size: 1 Each Price on request -
XIAP ligand-Linker Conjugate 2
SKU: QM-0013154 | Size: 1 Each Price on request -
XIAP ligand 5
SKU: QM-0013153 | Size: 1 Each Price on request -
XIAP ligand-Linker Conjugate 1
SKU: QM-0013149 | Size: 1 Each Price on request -
USP7 Ligand-Linker Conjugates 1
SKU: QM-0013083-01 | Size: 5 mg£1,412.02 GBP -
USP7 activator 1 [CAS 868940-26-5]
CAS: 868940-26-5 | SKU: QM-0011446-01 | Size: 5 mg£1,267.43 GBP -
VHL Ligand 36 [CAS 2250056-48-3]
CAS: 2250056-48-3 | SKU: QM-0011084 | Size: 1 Each Price on request -
VDR agonist 3
SKU: QM-0010210 | Size: 1 Each Price on request -
XPO1-ligand-1 [CAS 1076236-11-7]
CAS: 1076236-11-7 | SKU: QM-0009495 | Size: 1 Each Price on request -
Wnt pathway inhibitor 5 [CAS 1385817-77-5]
CAS: 1385817-77-5 | SKU: QM-0008977 | Size: 1 Each Price on request -
UMPK ligand 1 [CAS 1621866-83-8]
CAS: 1621866-83-8 | SKU: QM-0008942 | Size: 1 Each Price on request -
Wnt/β-catenin activator 1
SKU: QM-0008701 | Size: 1 Each Price on request -
WDR5 ligand 2 [CAS 2737222-78-3]
CAS: 2737222-78-3 | SKU: QM-0008544 | Size: 1 Each Price on request -
WRN inhibitor 13 [CAS 2923009-51-0]
CAS: 2923009-51-0 | SKU: QM-0008139 | Size: 1 Each Price on request -
VHL Ligand 38 [CAS 1360616-29-0]
CAS: 1360616-29-0 | SKU: QM-0004854 | Size: 1 Each Price on request -
Urotensin-II receptor antagonist-1 [CAS 1034708-07-0]
CAS: 1034708-07-0 | SKU: QM-0003152 | Size: 1 Each Price on request -
Wnt/β-catenin agonist 3 [CAS 912790-59-1]
CAS: 912790-59-1 | SKU: QM-0149522-01 | Size: 5 mg£124.00 GBP -
USP7/USP47 inhibitor [CAS 1247825-37-1]
CAS: 1247825-37-1 | SKU: QM-0144869-01 | Size: 5 mg£194.59 GBP -
WRN inhibitor 8 [CAS 3026502-95-1]
CAS: 3026502-95-1 | SKU: QM-0153042-01 | Size: 5 mg£928.45 GBP -
USP25/28 inhibitor AZ1 [CAS 2165322-94-9]
CAS: 2165322-94-9 | SKU: QM-0139145-01 | Size: 5 mg£118.38 GBP -
Wnt/β-catenin agonist 4 [CAS 912784-79-3]
CAS: 912784-79-3 | SKU: QM-0150559-01 | Size: 5 mg£118.38 GBP -
YAP/TAZ inhibitor-2 [CAS 2762617-31-0]
CAS: 2762617-31-0 | SKU: QM-0149350-01 | Size: 5 mg£363.47 GBP -
URAT1&XO inhibitor 2 [CAS 1239488-96-0]
CAS: 1239488-96-0 | SKU: QM-0151375-01 | Size: 5 mg£140.88 GBP -
WRN inhibitor 5 [CAS 2923009-95-2]
CAS: 2923009-95-2 | SKU: QM-0152031-01 | Size: 5 mg£381.69 GBP -
URAT1 inhibitor 1 [CAS 2268720-62-1]
CAS: 2268720-62-1 | SKU: QM-0138369-01 | Size: 5 mg£614.98 GBP