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A-381393 [CAS 726174-00-1]

A-381393 [CAS 726174-00-1]

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QM-0139033-01

£238.32 GBP
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Product Details

  • Description

    A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM) [1].

  • CAS Number

    [726174-00-1]

  • Molecular Formula

    C20H24N4

  • Molecular Weight

    320.43

  • Smiles

    CC1=CC=C(C=C1C)N2CCN(CC2)CC3=NC4=CC=CC=C4N3

  • Target

    Dopamine Receptor

  • Isoform

    5-HT2 Receptor; D3 Receptor; D4 Receptor

  • Purity

    99.92

  • Solubility

    DMSO : 51.67 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H315, H319

  • Precautions

    H315, H319
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Variant Variant total Quantity Price Variant total
5 mgQM-0139033-01
5 mgQM-0139033-01
£238.32/ea		 £0.00
£238.32/ea £0.00
10 mM - 1 mLQM-0139033-02
10 mM - 1 mLQM-0139033-02
£256.55/ea		 £0.00
£256.55/ea £0.00
10 mgQM-0139033-03
10 mgQM-0139033-03
£363.47/ea		 £0.00
£363.47/ea £0.00
25 mgQM-0139033-04
25 mgQM-0139033-04
£614.98/ea		 £0.00
£614.98/ea £0.00
50 mgQM-0139033-05
50 mgQM-0139033-05
£865.26/ea		 £0.00
£865.26/ea £0.00
100 mgQM-0139033-06
100 mgQM-0139033-06
£1,241.91/ea		 £0.00
£1,241.91/ea £0.00
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A-381393 [CAS 726174-00-1]

A-381393 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.