Ac-c[Cys-Glu-His-d-Phe-Arg-Trp-d-Cys]-Pro-Pro-Lys-Asp-NH2 [CAS 596135-92-1]

Ac-c[Cys-Glu-His-d-Phe-Arg-Trp-d-Cys]-Pro-Pro-Lys-Asp-NH2 (compound 5) is a selective hMC5R antagonist ligand with an IC50 of 10 nM[1].

[596135-92-1]

C65H89N19O16S2

1456.65

O=C(N[C@H](CSSC[C@@H](C(N[C@H](C(N[C@H](C(N[C@@H](C(N[C@H](C(N1)=O)CCCNC(N)=N)=O)CC2=CC=CC=C2)=O)CC3=CN=CN3)=O)CCC(O)=O)=O)NC(C)=O)C(N4[C@@H](CCC4)C(N5[C@@H](CCC5)C(N[C@@H](CCCCN)C(N[C@H](C(N)=O)CC(O)=O)=O)=O)=O)=O)[C@@H]1CC6=CNC7=CC=CC=C67

Melanocortin Receptor

MC5R

Room temperature