ADAR1-IN-1 [CAS 2734853-87-1]

ADAR1-IN-1 is a potent ADAR1 inhibitor. ADAR1-IN-1 significantly suppressed DU-145 cell proliferation (IC50 = 1.11 μM), clonogenicity, migration, and invasion, arrests cell cycle, and induces apoptosis. ADAR1-IN-1 safely and effectively inhibits tumor growth. ADAR1-IN-1 can be used for the study of prostate cancer (PCa) [1].

[2734853-87-1]

C17H15F4N5O6S

493.39

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Adenosine Deaminase; Apoptosis

Room temperature