[Ala1, 3, 11, 15]-Endothelin (53-63) (TFA)

[Ala1,3,11,15]-Endothelin (53-63) (TFA) is an ETB agonist. [Ala1,3,11,15]-Endothelin (53-63) (TFA) has selectivity for ETB with IC50 values range from 0.33 nM to 0.61 nM. [Ala1,3,11,15]-Endothelin (53-63) (TFA) can be used for the research of vasoconstriction[1].

C111H164F3N25O34S

2481.7

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Endothelin Receptor

ETB

10 mM in DMSO

Room temperature