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Aprocitentan [CAS 1103522-45-7]

Aprocitentan [CAS 1103522-45-7]

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QM-0076157-01

£118.38 GBP
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Product Details

  • Description

    Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is an orally active dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively. Aprocitentan is an antihypertensive agent[1].

  • CAS Number

    [1103522-45-7]

  • Molecular Formula

    C16H14Br2N6O4S

  • Molecular Weight

    546.19

  • Smiles

    O=S(N)(NC1=NC=NC(OCCOC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O

  • Target

    Endothelin Receptor

  • Isoform

    ETA; ETB

  • Purity

    99.55

  • Solubility

    DMSO : 25 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H315, H319, H335

  • Precautions

    H302, H315, H319, H335
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Variant Variant total Quantity Price Variant total
1 mgQM-0076157-01
1 mgQM-0076157-01
£118.38/ea		 £0.00
£118.38/ea £0.00
5 mgQM-0076157-02
5 mgQM-0076157-02
£297.86/ea		 £0.00
£297.86/ea £0.00
10 mM - 1 mLQM-0076157-03
10 mM - 1 mLQM-0076157-03
£347.68/ea		 £0.00
£347.68/ea £0.00
10 mgQM-0076157-04
10 mgQM-0076157-04
£407.21/ea		 £0.00
£407.21/ea £0.00
25 mgQM-0076157-05
25 mgQM-0076157-05
£673.29/ea		 £0.00
£673.29/ea £0.00
50 mgQM-0076157-06
50 mgQM-0076157-06
£923.59/ea		 £0.00
£923.59/ea £0.00
100 mgQM-0076157-07
100 mgQM-0076157-07
£1,229.77/ea		 £0.00
£1,229.77/ea £0.00
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Aprocitentan [CAS 1103522-45-7]

Aprocitentan is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.