CBP/p300-IN-5 [CAS 1889284-33-6]

P300/CBP-IN-5 is a potent p300/CBP histone acetyltransferase inhibitor extracted from patent WO2016044770A1, Example 715, has an IC50 of 18.8 nM[1].

[1889284-33-6]

C29H27F5N6O4

618.55

O=C(CN(C1=O)C(N[C@@]21C[C@H](C3=C2C=CC(C4=CN(N=C4)CC(NC)=O)=C3)F)=O)N([C@H](C(F)(F)F)C)CC5=CC=C(C=C5)F

Histone Acetyltransferase

CBP/p300

97

DMSO : 60 mg/mL (ultrasonic; warming)

-20°C, 3 years (Powder)

Blue Ice