ChemR23-IN-1 [CAS 2378640-10-7]

ChemR23-IN-1 (compound 2) is a ChemR23 inhibitor with IC50s of 38 nM and 100 nM for human and mouse ChemR23, respectively. ChemR23-IN-1 inhibits chemotaxis of CAL-1 triggered by Chemerin in vitro[1].

[2378640-10-7]

C28H29N7O2

495.58

C[C@@H](N(CCCC)C1=NC2=CC(C(NC)=O)=CC=C2O1)C3=CC=C(C4=CC=CC=C4C5=NN=NN5)C=C3

Chemerin Receptor

98.82

DMSO : 100 mg/mL (ultrasonic)

-20°C, 3 years; 4°C, 2 years (Powder)

Room Temperature