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CK2/ERK8-IN-1 [CAS 1085822-09-8]
CK2/ERK8-IN-1 [CAS 1085822-09-8]
SKU:QM-0145275-01
£78.82 GBP
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![CK2/ERK8-IN-1 [CAS 1085822-09-8]](http://quantimol.com/cdn/shop/files/quantimol-021.png?v=1773515276&width=1445)
Product Details
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Description
CK2/ERK8-IN-1 is a dual casein kinase 2 (CK2) (Ki of 0.25 μM) and ERK8 (MAPK15, ERK7) inhibitor with IC50s of 0.50 μM. CK2/ERK8-IN-1 also binds to PIM1, HIPK2 (homeodomain-interacting protein kinase 2), and DYRK1A with Kis of 8.65 μM, 15.25 μM, and 11.9 μM, respectively. CK2/ERK8-IN-1 has pro-apoptotic efficacy[1].
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CAS Number
[1085822-09-8]
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Molecular Formula
C11H9Br4N3O2
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Molecular Weight
534.82
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Smiles
O=C(O)CN1C2=C(Br)C(Br)=C(Br)C(Br)=C2N=C1N(C)C
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Target
Apoptosis; Casein Kinase; DYRK; ERK; Pim
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Isoform
CK2; DYRK1; ERK8; PIM1
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Concentration
10mM
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Purity
99
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Solubility
DMSO : 16.67 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years (Powder)
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Shipping Conditions
Blue Ice
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CK2/ERK8-IN-1 [CAS 1085822-09-8]
CK2/ERK8-IN-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.