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(E/Z) -GSK5182 [CAS 2699724-40-6]
(E/Z) -GSK5182 [CAS 2699724-40-6]
SKU:QM-0136965-01
£323.38 GBP
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![(E/Z) -GSK5182 [CAS 2699724-40-6]](http://quantimol.com/cdn/shop/files/quantimol-021.png?v=1773515276&width=1445)
Product Details
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Description
(E/Z) -GSK5182 is a racemic compound of (E) -GSK5182 and (Z) -GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3].
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CAS Number
[2699724-40-6]
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Molecular Formula
C27H31NO3
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Molecular Weight
417.54
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Smiles
OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)OCCN(C)C)\C3=CC=C(C=C3)O
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Target
Estrogen Receptor/ERR; Reactive Oxygen Species (ROS)
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Purity
98.9
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Solubility
DMSO : ≥ 75 mg/mL
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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(E/Z) -GSK5182 [CAS 2699724-40-6]
(E/Z) -GSK5182 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.