Endomorphin 1 [CAS 189388-22-5]

Endomorphin 1, a high affinity, highly selective agonist of the μ-opioid receptor (Ki: 1.11 nM), displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin 1 has antinociceptive properties[1][2][4].

[189388-22-5]

C34H38N6O5

610.7

O=C(N)[C@H](CC1=CC=CC=C1)NC([C@H](CC2=CNC3=CC=CC=C23)NC([C@H]4N(C([C@H](CC5=CC=C(C=C5)O)N)=O)CCC4)=O)=O

Opioid Receptor

μ Opioid Receptor/MOR

99.92

DMSO : ≥ 50 mg/mL

-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light, under nitrogen)

Blue Ice

H302, H315, H319, H335

H302, H315, H319, H335