EPZ-4777 [CAS 1381761-52-9]

EPZ-4777 is a selective DOT1L inhibitor which inhibits H3K79 methylation in cancer cells, blocks the expression of leukemogenic genes, and selectively kills cells that contain the translocation. EPZ-4777 can be used for cancer research[1].

[1381761-52-9]

C27H40N8O4

540.66

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Histone Methyltransferase

Room temperature