Estrone-N-O-C1-amido [CAS 138219-84-8]

Estrone-N-O-C1-amido (ERα ligand 1) is an Estrone-based estrogen ligand, which targets estrogen receptor α (ERα) . Estrone-N-O-C1-amido (ERα ligand 1) binds to cIAP1 ligand Bestatin via a linker to form SNIPER[1].

[138219-84-8]

C20H26N2O3

342.43

O=C(N)CO/N=C1CC[C@]2([H])[C@]\1(C)CC[C@@]3([H])[C@@]2([H])CCC4=C3C=CC(O)=C4

Estrogen Receptor/ERR; Ligands for Target Protein for PROTAC

10 mM in DMSO

Room temperature