FGA146

FGA146 is a dual, selective inhibitor for Mpro and human Cathepsin L, with Kis of 2.19 μM, 0.96 μM and 0.87 μM, for Mal-Mpro, pET21-Mpro and Cathepsin L, respectively. FGA146 reveals an antiviral activity against SARS-CoV-2[1].

C24H31N5O6

485.53

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Cathepsin; Virus Protease

Cathepsin L

10 mM in DMSO

Room temperature