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Fmoc-L-Asn (EDA-N3) -OH [CAS 2616562-74-2]

Fmoc-L-Asn (EDA-N3) -OH [CAS 2616562-74-2]

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SKU:QM-0069656

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  • Description

    Fmoc-L-Asn (EDA-N3) -OH is a click chemistry reagent containing an azide group. This building block is reported in literature for the modification of Amanitin via Click Chemistry. Alpha-Amanitin is the deadliest member of the amatoxin peptide family produced by the death-cap mushroom A. phalloides. It is an orally available, rigid, bicyclic octapeptide and one of the most lethal known natural products (LD50 = 50-100 μg/kg) acting as highly selective allosteric inhibitor of the RNA polymerase II[1]. It contains an azide group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing alkyne groups. It can also undergo ring strain-promoted alkyne-azide cycloaddition (SPAAC) with molecules containing DBCO or BCN groups.

  • CAS Number

    [2616562-74-2]

  • Molecular Formula

    C21H21N5O5

  • Molecular Weight

    423.42

  • Smiles

    [N-]=[N+]=NCCNC(C[C@@H](C(O)=O)NC(OCC1C2=CC=CC=C2C3=CC=CC=C31)=O)=O

  • Target

    ADC Linker

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature

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Fmoc-L-Asn (EDA-N3) -OH [CAS 2616562-74-2]

Fmoc-L-Asn (EDA-N3) -OH is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.