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Gamcemetinib [CAS 1887069-10-4]

Gamcemetinib [CAS 1887069-10-4]

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QM-0146722-01

£238.32 GBP
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Product Details

  • Description

    Gamcemetinib (CC-99677) is a potent, covalent, and irreversible inhibitor of the mitogen-activated protein (MAP) kinase-activated protein kinase-2 (MK2) pathway in both biochemical (IC50=156.3 nM) and cell based assays (EC50=89 nM) . Gamcemetinib is extracted from patent WO2020236636, compound 1[1].

  • CAS Number

    [1887069-10-4]

  • Molecular Formula

    C22H20ClN5O3S

  • Molecular Weight

    469.94

  • Smiles

    O=C1C2=C(NC[C@H](N1)C)C3=C(S2)C=CC4=NC(OC5=NC(Cl)=NC=C5COCC)=CC=C34

  • Target

    MAPKAPK2 (MK2)

  • Concentration

    10mM

  • Purity

    99.06

  • Solubility

    DMSO : 37.5 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
1 mgQM-0146722-01
1 mgQM-0146722-01
£238.32/ea		 £0.00
£238.32/ea £0.00
5 mgQM-0146722-02
5 mgQM-0146722-02
£452.17/ea		 £0.00
£452.17/ea £0.00
10 mM - 1 mLQM-0146722-03
10 mM - 1 mLQM-0146722-03
£465.53/ea		 £0.00
£465.53/ea £0.00
10 mgQM-0146722-04
10 mgQM-0146722-04
£740.12/ea		 £0.00
£740.12/ea £0.00
25 mgQM-0146722-05
25 mgQM-0146722-05
£1,279.58/ea		 £0.00
£1,279.58/ea £0.00
50 mgQM-0146722-06
50 mgQM-0146722-06
£1,681.74/ea		 £0.00
£1,681.74/ea £0.00
100 mgQM-0146722-07
100 mgQM-0146722-07
£2,309.90/ea		 £0.00
£2,309.90/ea £0.00
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Gamcemetinib [CAS 1887069-10-4]

Gamcemetinib is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.