GluN1/3A-IN-1 [CAS 1147526-22-4]

GluN1/3A-IN-1 (Compound GM-10) is a GluN1/GluN3A NMDA receptor inhibitor. GluN1/3A-IN-1 exhibits potent inhibitory activity against GluN1/GluN3A (IC50: 0.98 µM) . GluN1/3A-IN-1 exerts its inhibitory effect by targeting the pre-M1 region and forming hydrogen bond interactions with key residues. GluN1/3A-IN-1 can be used to study GluN1/GluN3A-related neurological diseases[1].

[1147526-22-4]

C23H17NO5

387.38

O=C(C1=C(C=C(C=C1)O)O)OCC(C2C(C3=CC=CC=C3)=NC4=C2C=CC=C4)=O

IGluR

98.06

-20°C, 3 years (Powder)

Blue Ice