GR 250495X [CAS 192057-17-3]

GR 250495X is an inhaled glucocorticoid receptor agonist. GR 250495X is designed as a antedrug, which takes effect locally in the lungs but is rapidly metabolized and inactivated in the bloodstream after entering the systemic circulation, thereby minimizing systemic side effects. GR 250495X can be used in asthma research[1].

[192057-17-3]

C28H36F2O7S

554.64

O=C(OCC1)[C@H]1SC([C@]23[C@@]4([C@@]([C@@]5([H])[C@]([C@H](C4)O)([C@@]6(C([C@H](C5)F)=CC(CC6)=O)C)F)([H])C[C@@]2([H])O[C@H](O3)CCC)C)=O

Glucocorticoid Receptor

Room temperature