Name: GRK5-IN-2 [CAS 1642839-27-7]
Brand: QuantiMol
SKU: QM-0145640-01
Price: 135.25 GBP
Availability: InStock

Product Details

Description
GRK5-IN-2 (compound 707), a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 of 49.7 μM. GRK5-IN-2 regulates the expression and/or release of insulin and is useful for the metabolic disease research[1][2].
CAS Number
[1642839-27-7]
Molecular Formula
C20H20N4O4
Molecular Weight
380.4
Smiles
COC1=C(OC)C(OC)=CC(NC2=CC3=C(N=C(C4=CC=CO4)N3C)C=N2)=C1
Target
ERK; G Protein-coupled Receptor Kinase (GRK)
Purity
99.91
Solubility
DMSO : 62.5 mg/mL (ultrasonic; warming; heat to 60°C)
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Shipping Conditions
Room Temperature

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Variant	Variant total	Quantity	Price	Variant total
5 mgQM-0145640-01	5 mgQM-0145640-01 £135.25/ea	£0.00	Quantity	£135.25/ea	£0.00

10 mM - 1 mLQM-0145640-02	10 mM - 1 mLQM-0145640-02 £146.50/ea	£0.00	Quantity	£146.50/ea	£0.00

10 mgQM-0145640-03	10 mgQM-0145640-03 £238.32/ea	£0.00	Quantity	£238.32/ea	£0.00

25 mgQM-0145640-04	25 mgQM-0145640-04 £426.65/ea	£0.00	Quantity	£426.65/ea	£0.00

50 mgQM-0145640-05	50 mgQM-0145640-05 £652.64/ea	£0.00	Quantity	£652.64/ea	£0.00

100 mgQM-0145640-06	100 mgQM-0145640-06 £1,015.92/ea	£0.00	Quantity	£1,015.92/ea	£0.00

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GRK5-IN-2 [CAS 1642839-27-7]

GRK5-IN-2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.