GRL-098-22

GRL-098-22 (Compound 6t) is a potent inhibitor targeting G protein-coupled receptor kinase 5 (GRK5) and GRK6 with IC50 values of 0.6 μM and 0.19 μM, respectively. GRL-098-22 is promising for research of diseases such as heart failure and multiple myeloma[1].

C34H39FN6O5

630.71

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G Protein-coupled Receptor Kinase (GRK)

Room temperature