GSK256073 [CAS 862892-90-8]
GSK256073 [CAS 862892-90-8]
SKU:QM-0139551-01
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Product Details
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Description
GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2) . GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM) and dyslipidemia[1][2]. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
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CAS Number
[862892-90-8]
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Molecular Formula
C10H13ClN4O2
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Molecular Weight
256.69
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Smiles
O=C(N(C1=C2NC(Cl)=N1)CCCCC)NC2=O
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Target
GPR109A
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Concentration
10mM
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Purity
99.39
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Solubility
DMSO : 16.67 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H361
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Precautions
H302, H361
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GSK256073 [CAS 862892-90-8]
GSK256073 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.