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GSK256073 (tris) [CAS 1228650-42-7]

GSK256073 (tris) [CAS 1228650-42-7]

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SKU:QM-0098568

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  • Description

    GSK256073 tris is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2) . GSK256073 tris acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM) and dyslipidemia[1][2]. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2

  • CAS Number

    [1228650-42-7]

  • Molecular Formula

    C14H24ClN5O5

  • Molecular Weight

    377.82

  • Smiles

    O=C1NC(N(CCCCC)C2=C1NC(Cl)=N2)=O.OCC(CO)(CO)N

  • Target

    GPR109A

  • Shipping Conditions

    Room temperature

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GSK256073 (tris) [CAS 1228650-42-7]

GSK256073 (tris) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.