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GSK2801 [CAS 1619994-68-1]
GSK2801 [CAS 1619994-68-1]
SKU:QM-0152029-01
£127.38 GBP
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Product Details
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Description
GSK2801, a chemical probe, is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4[1].
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CAS Number
[1619994-68-1]
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Molecular Formula
C20H21NO4S
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Molecular Weight
371.45
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Smiles
O=C(C)C1=CC(C2=C(S(=O)(C)=O)C=CC=C2)=C3N1C=CC(OCCC)=C3
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Target
Apoptosis; Epigenetic Reader Domain
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Purity
99.95
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Solubility
DMSO : 50 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H315, H319, H335
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Precautions
H302, H315, H319, H335
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GSK2801 [CAS 1619994-68-1]
GSK2801 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.