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GSK6853 [CAS 1910124-24-1]
GSK6853 [CAS 1910124-24-1]
SKU:QM-0079163-01
£78.82 GBP
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![GSK6853 [CAS 1910124-24-1]](http://quantimol.com/cdn/shop/files/quantimol-021.png?v=1773515276&width=1445)
Product Details
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Description
GSK6853, a chemical probe, is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd = 9.5) and greater than 1600-fold selectivity over all other bromodomains[1].
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CAS Number
[1910124-24-1]
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Molecular Formula
C22H27N5O3
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Molecular Weight
409.48
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Smiles
C[C@@H]1CNCCN1C2=C(NC(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O
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Target
Epigenetic Reader Domain
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Purity
99.89
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Solubility
DMSO : 25 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H315, H319, H335
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Precautions
H302, H315, H319, H335
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GSK6853 [CAS 1910124-24-1]
GSK6853 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.