GSK837149A [CAS 13616-29-0]
GSK837149A [CAS 13616-29-0]
SKU:QM-0139252-01
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Product Details
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Description
GSK837149A is a selective inhibitor of human Fatty Acid Synthase (FASN) targeting the KR domain. GSK837149A has reversible inhibition effect on FASN and selectivity for type I FASN (Ki=30 nM) . GSK837149A is also a competitive inhibitor of NADPH and a non-competitive inhibitor of acetoacetyl-CoA. GSK837149A can be used for the research of obesity and breast cancer[1][2].
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CAS Number
[13616-29-0]
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Molecular Formula
C23H22N8O5S2
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Molecular Weight
554.6
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Smiles
O=C(NC1=CC=C(C=C1)S(=O)(NC2=NC=CC(C)=N2)=O)NC3=CC=C(C=C3)S(=O)(NC4=NC=CC(C)=N4)=O
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Target
Fatty Acid Synthase (FASN)
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Purity
99
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Solubility
DMSO : 10 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Hazard Statement
H319
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Precautions
H319
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GSK837149A [CAS 13616-29-0]
GSK837149A is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.