HSR-IN-1

HSR-IN-1 (Compound 28) is an effective hSR (human serine racemase) inhibitor. In the presence of the cofactor Pyridoxal 5'-phosphate monohydrate , HSR-IN-1 has a Kd value of 5.4 μM and an IC50 of 18.3 μM for hSR, while the IC50 of HSR-IN-1 alone is 4.7 μM. HSR-IN-1 can be used for research on central nervous system diseases[1].

C15H16ClNO3

293.75

[NH3+]OC(C(O)=O)CC1=CC=C(C2=CC=CC=C2)C=C1.[Cl-]

Serine Racemase (SR)

Room temperature