Human enteropeptidase-IN-1 [CAS 1802891-20-8]

Human enteropeptidase-IN-1 (compound 6b) is a highly potent, orally active and low systemic exposure enteropeptidase inhibitor. Human enteropeptidase-IN-1 boosts the increase in fecal protein output, and exhibits potent body weight loss in diet-induced obese (DIO) rat model. Human enteropeptidase-IN-1 can be used for anti-obesity research[1].

[1802891-20-8]

C20H18N4O7

426.38

OC(C[C@]1(CC(C2=CC(OC(C3=CC=C(C=C3)NC(N)=N)=O)=CC=C2)=NO1)C(O)=O)=O

Enteropeptidase

10 mM in DMSO

Room temperature