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HYL001 [CAS 2426547-83-1]

HYL001 [CAS 2426547-83-1]

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SKU:QM-0119124-01

£129.63 GBP
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  • Description

    HYL001 (compund 338) is a potent inhibitor of TGFβ receptor 1 (ALK5) that is approximately 9 times more potent than the structurally related compound Galunisertib and is able to eliminate liver metastases established in mice[1].

  • CAS Number

    [2426547-83-1]

  • Molecular Formula

    C21H18N4O

  • Molecular Weight

    342.39

  • Smiles

    OC1=CC2=C(C3=C(CCC4)N4N=C3C5=CC=CC(C)=N5)C=CN=C2C=C1

  • Target

    TGF-β Receptor

  • Purity

    99.94

  • Solubility

    DMSO : 17.5 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

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Variant Variant total Quantity Price Variant total
5 mgQM-0119124-01
5 mgQM-0119124-01
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£83.70
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£129.63/ea
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£83.70
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£129.63/ea
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10 mM - 1 mLQM-0119124-02
10 mM - 1 mLQM-0119124-02
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£91.80
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£139.75/ea
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£91.80
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10 mgQM-0119124-03
10 mgQM-0119124-03
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£134.10
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£231.03/ea
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£134.10
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£231.03/ea
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25 mgQM-0119124-04
25 mgQM-0119124-04
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£270.00
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£414.50/ea
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£270.00
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50 mgQM-0119124-05
50 mgQM-0119124-05
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£431.10
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£631.99/ea
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£431.10
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£631.99/ea
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100 mgQM-0119124-06
100 mgQM-0119124-06
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£687.60
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£978.26/ea
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£687.60
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£978.26/ea
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HYL001 [CAS 2426547-83-1]

HYL001 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.