L-798106 [CAS 244101-02-8]

L-798106 is potent and highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM), it also has micromolar activities at the EP4, EP1 and EP2 receptors with Ki values of 916 nM, >5000 nM and >5000 nM, respectively[1].

[244101-02-8]

C27H22BrNO4S

536.44

O=C(NS(=O)(C1=CC(Br)=CC=C1OC)=O)/C=C/C2=CC=CC=C2CC3=CC=C4C=CC=CC4=C3

Prostaglandin Receptor

EP

99.91

10 mM in DMSO

-20°C, 3 years (Powder)

Blue Ice

H413

P273-P501