L-803087 [CAS 217480-26-7]

L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM. L-803087 is >280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice[1][2].

[217480-26-7]

C25H29F2N5O3

485.53

N=C(N)NCCC[C@@H](C(OC)=O)NC(CCCC1=C(C2=CC=CC=C2)NC3=C1C=C(F)C=C3F)=O

Somatostatin Receptor

99.66

DMSO : 250 mg/mL (ultrasonic)

-20°C, 3 years (Powder)

Blue Ice