Melengestrol acetate-d6

Melengestrol acetate-d6 is the deuterium labeled Melengestrol acetate. Melengestrol acetate is a progesterone derivative, acts as an orally active corticosteroid hormone to promote endometrial proliferation, pregnancy maintenance, and delay of menstrual activity[1]. Melengestrol Acetate is used as a contraceptive agent for growth promoting effects and suppression of estrus in animals. Melengestrol acetate inhibits both the androgen-dependent and -independent prostatic tumors in vivo and can be used for cancer research[2].

C25H26D6O4

402.56

C[C@]1([C@](C2)([H])[C@]3([H])C=C(C)C4=C([2H])C(C([2H])([2H])C[C@]4(C)[C@@]3([H])CC1)=O)[C@](C(C([2H])([2H])[2H])=O)(OC(C)=O)C2=C

Isotope-Labeled Compounds; Progesterone Receptor

10 mM in DMSO

Room temperature