MRS2365 (trisodium)

MRS2365 trisodium is a potent and selective P2Y1 receptor (EC50=0.4 nM) /[35S]GTPγS binding/β-arrestin 2 recruitment agonist. MRS2365 trisodium relieves mechanical allodynia and increases mechanical sensitivity[1][2][3][4].

C13H16N5Na3O9P2S

549.28

O=P(OP(O[Na])(O[Na])=O)(O[Na])OC[C@]12[C@@H](O)[C@@H](O)[C@H](N3C=NC4=C(N)N=C(SC)N=C34)[C@@]1([H])C2

Arrestin; P2Y Receptor

P2Y1 Receptor

10 mM * 182 μL in Water

99

10 mM in DMSO

Solution, -20°C, 2 years

Blue Ice