MRS8209

MRS8209 is the antagonist for serotonin receptor with a Ki of 4.27 nM for 5-HT2BR. MRS8209 exhibits protective effect on pressure at airway opening (PAO), and can be used in research of pulmonary fibrosis[1].

C17H19IN6O2

466.28

O[C@@H]1[C@H](O)[C@@]2(C#N)[C@H](C2)[C@H]1N3C(N=C(I)N=C4NC5CCCC5)=C4N=C3

5-HT Receptor

α-1 microglobulin

Room temperature