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Multi-kinase-IN-6 [CAS 3009081-73-3]

Multi-kinase-IN-6 [CAS 3009081-73-3]

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SKU:QM-0072412

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  • Description

    Multi-kinase-IN-6 (compound 10e) is a multikinase inhibitor that shows good enzyme inhibitory activity against TrkA, ALK2, c-KIT, EGFR, PIM1, CK2α, CHK1, and CDK2. Multi-kinase-IN-6 reveals antiproliferative activity against MCF7, HCT116 and EKVX with IC50 values of 3.36 μM, 1.40 μM and 3.49 μM, respectively. Multi-kinase-IN-6 shows cell cycle arrest at the G1/S phase and G1 phase in MCF7 and HCT116 cells with good apoptotic effect[1].

  • CAS Number

    [3009081-73-3]

  • Molecular Formula

    C17H15N5O2

  • Molecular Weight

    321.33

  • Smiles

    COC(C=C1)=CC=C1C2=CC=NC3=C(C4=NOC(C)=N4)C(C)=NN32

  • Target

    Anaplastic lymphoma kinase (ALK) ; Apoptosis; Casein Kinase; CDK; Checkpoint Kinase (Chk) ; c-Kit; EGFR; Pim; Trk Receptor

  • Isoform

    CDK2; Chk1; CK2; EGFR/ErbB1/HER1; PIM1; TrkA

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature

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Multi-kinase-IN-6 [CAS 3009081-73-3]

Multi-kinase-IN-6 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.