1 1

NBI-42902 [CAS 352290-60-9]

NBI-42902 [CAS 352290-60-9]

Size

QM-0145810-01

£532.36 GBP
Sale Sold out

Request quote or documents

View full details

Product Details

  • Description

    NBI-42902 is an orally active, potent functional and competitive antagonist of GnRH receptor with an IC50 value of 0.79 nM, a Ki value of 0.56 nM, respectively. NBI-42902 inhibits GnRH-stimulated inositol phosphate (IP) accumulation, Ca2+ flux, and ERK1/2 activation. NBI-42902 inhibits serum luteinizing hormone (LH) in castrated male macaques. NBI-42902 can be used for research on sex-hormone-related diseases[1].

  • CAS Number

    [352290-60-9]

  • Molecular Formula

    C27H24F3N3O3

  • Molecular Weight

    495.49

  • Smiles

    O=C1N(C[C@H](N)C2=CC=CC=C2)C(C(C3=CC=CC(OC)=C3F)=C(C)N1CC4=C(F)C=CC=C4F)=O

  • Target

    GnRH Receptor; PERK

  • Concentration

    10mM

  • Purity

    98.65

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H315, H319, H335

  • Precautions

    H302, H315, H319, H335
Learn more
Variant Variant total Quantity Price Variant total
5 mgQM-0145810-01
5 mgQM-0145810-01
£532.36/ea		 £0.00
£532.36/ea £0.00
10 mM - 1 mLQM-0145810-02
10 mM - 1 mLQM-0145810-02
£576.10/ea		 £0.00
£576.10/ea £0.00
10 mgQM-0145810-03
10 mgQM-0145810-03
£821.52/ea		 £0.00
£821.52/ea £0.00
25 mgQM-0145810-04
25 mgQM-0145810-04
£1,668.38/ea		 £0.00
£1,668.38/ea £0.00
50 mgQM-0145810-05
50 mgQM-0145810-05
£2,637.95/ea		 £0.00
£2,637.95/ea £0.00
100 mgQM-0145810-06
100 mgQM-0145810-06
£4,191.94/ea		 £0.00
£4,191.94/ea £0.00
View cart
0

Total items

£0.00

Product subtotal

Taxes, discounts and shipping calculated at checkout.
View cart

Related Products

Other industry favorites

NBI-42902 [CAS 352290-60-9]

NBI-42902 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.