OMDM-5 [CAS 616884-66-3]

OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM) [1].

[616884-66-3]

C26H44N2O3

432.64

CCCCCCCC/C=C\CCCCCCCC(NNCC1=CC=C(O)C(OC)=C1)=O

Endogenous Metabolite; TRP Channel

10 mM in DMSO

Room temperature