[Orn5]-URP (TFA)

[Orn5]-URP TFA is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP TFA displays no agonist activity[1][2].

C48H62N10O10S2.xC2HF3O2

OC(C(F)(F)F)=O.O=C([C@@H](NC([C@H](CSSC[C@H](NC([C@@H](NC([C@@H](NC1=O)CCCN)=O)CC2=CC=C(C=C2)O)=O)C(N[C@H](C(O)=O)C(C)C)=O)NC([C@@H](N)C)=O)=O)CC3=CC=CC=C3)N[C@H]1CC4=CNC5=CC=CC=C45

Urotensin Receptor

H2O

Room temperature