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Orvepitant (maleate) [CAS 579475-24-4]

Orvepitant (maleate) [CAS 579475-24-4]

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QM-0077999-01

£301.50 GBP
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Product Details

  • Description

    Orvepitant maleate (GW823296 maleate) is potent, selective, orally active and well-tolerated neurokinin-1 receptor (NK-1) antagonist with a pKi of 10.2 for human neurokinin-1 receptor. Orvepitant maleate can across the blood-brain barrier. Orvepitant maleate has the potential for depressive disorder and chronic refractory cough (CRC) treatment[1][2].

  • CAS Number

    [579475-24-4]

  • Molecular Formula

    C35H39F7N4O6

  • Molecular Weight

    744.7

  • Smiles

    O=C(N1[C@@H](C2=CC=C(F)C=C2C)C[C@@H](N3C[C@@](CCC4=O)([H])N4CC3)CC1)N([C@@H](C5=CC(C(F)(F)F)=CC(C(F)(F)F)=C5)C)C.O=C(O)/C=C\C(O)=O

  • Target

    Neurokinin Receptor

  • Isoform

    NK1R

  • Concentration

    10mM

  • Purity

    99.99

  • Solubility

    DMSO : 30 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H361

  • Precautions

    H302, H361
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Variant Variant total Quantity Price Variant total
5 mgQM-0077999-01
5 mgQM-0077999-01
£301.50/ea		 £0.00
£301.50/ea £0.00
10 mM - 1 mLQM-0077999-02
10 mM - 1 mLQM-0077999-02
£461.88/ea		 £0.00
£461.88/ea £0.00
10 mgQM-0077999-03
10 mgQM-0077999-03
£489.83/ea		 £0.00
£489.83/ea £0.00
25 mgQM-0077999-04
25 mgQM-0077999-04
£928.45/ea		 £0.00
£928.45/ea £0.00
50 mgQM-0077999-05
50 mgQM-0077999-05
£1,430.24/ea		 £0.00
£1,430.24/ea £0.00
100 mgQM-0077999-06
100 mgQM-0077999-06
£2,121.57/ea		 £0.00
£2,121.57/ea £0.00
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Orvepitant (maleate) [CAS 579475-24-4]

Orvepitant (maleate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.