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P300 bromodomain-IN-1
P300 bromodomain-IN-1
SKU:QM-0066877
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Quantity
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Product Details
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Description
P300 bromodomain-IN-1 (Compoun 1u) is a potent p300 (EP300) bromodomain inhibitor with an IC50 of 49 nM. P300 bromodomain-IN-1 suppresses the expression of c-Myc and induces G1/G0 phase arrest and apoptosis in OPM-2 cells[1].
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Molecular Formula
C29H31ClN4O4
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Molecular Weight
535.03
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Smiles
COC1=CC=C(C=C1Cl)N2C(C[C@H]2C3=NC4=CC(C5=C(ON=C5C)C)=CC=C4N3[C@H]6CC[C@@H](CC6)OC)=O
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Target
Epigenetic Reader Domain; Histone Acetyltransferase
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Isoform
CBP/p300
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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P300 bromodomain-IN-1
P300 bromodomain-IN-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.