Pan-HER-IN-2 [CAS 1639040-95-1]

Name: Pan-HER-IN-2 [CAS 1639040-95-1]
Brand: QuantiMol
SKU: QM-0148324-01
Price: 382.91 GBP
Availability: InStock

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SKU:QM-0148324-01

£382.91 GBP

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Product Details

Description
Pan-HER-IN-2 (Compound C6) is a reversible, orally active pan-HER inhibitor with IC50 values of 0.72, 2.0, 8.2 and 75.1 nM against EGFR, HER4, EGFRT790M/L858R and HER2, respectively. pan-HER-IN-2 induces apoptosis and shows antitumor activities[1].
CAS Number
[1639040-95-1]
Molecular Formula
C19H15BrClN5O
Molecular Weight
444.71
Smiles
O=C(NC1=CC=C2N=CN=C(C2=C1)NC3=CC4=C(NC=C4Br)C=C3)CCCl
Target
Apoptosis; EGFR
Isoform
EGFR/ErbB1/HER1; ErbB2/HER2; ErbB4/HER4
Purity
98.1
Solubility
DMSO : 100 mg/mL (ultrasonic)
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Shipping Conditions
Room Temperature

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Variant	Variant total	Quantity	Price	Variant total
5 mgQM-0148324-01	5 mgQM-0148324-01 £382.91/ea	£0.00	Quantity	£382.91/ea	£0.00

10 mgQM-0148324-02	10 mgQM-0148324-02 £583.38/ea	£0.00	Quantity	£583.38/ea	£0.00

25 mgQM-0148324-03	25 mgQM-0148324-03 £1,116.77/ea	£0.00	Quantity	£1,116.77/ea	£0.00

50 mgQM-0148324-04	50 mgQM-0148324-04 £1,744.92/ea	£0.00	Quantity	£1,744.92/ea	£0.00

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Pan-HER-IN-2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.