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PBRM1-BD2-IN-5 [CAS 2819989-61-0]

PBRM1-BD2-IN-5 [CAS 2819989-61-0]

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SKU:QM-0150563-01

£351.32 GBP
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  • Description

    PBRM1-BD2-IN-5 is a potent PBRM1 Bromodomain inhibitor with Kd values of 1.5 μM and 3.9 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.26 μM for PBRM1-BD2. PBRM1-BD2-IN-5 reduces the binding of full-length PBRM1 within the PBAF complex in cell lysates to acetylated histone peptide. PBRM1-BD2-IN-5 can be used to research anticancer[1].

  • CAS Number

    [2819989-61-0]

  • Molecular Formula

    C15H13ClN2O

  • Molecular Weight

    272.73

  • Smiles

    O=C1NC(C2=CC=CC(C)=C2)NC3=C1C(Cl)=CC=C3

  • Target

    Epigenetic Reader Domain

  • Purity

    99.75

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

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Variant Variant total Quantity Price Variant total
5 mgQM-0150563-01
5 mgQM-0150563-01
£351.32/ea
£0.00
£351.32/ea £0.00
10 mM - 1 mLQM-0150563-02
10 mM - 1 mLQM-0150563-02
£381.69/ea
£0.00
£381.69/ea £0.00
10 mgQM-0150563-03
10 mgQM-0150563-03
£489.83/ea
£0.00
£489.83/ea £0.00
25 mgQM-0150563-04
25 mgQM-0150563-04
£777.78/ea
£0.00
£777.78/ea £0.00
50 mgQM-0150563-05
50 mgQM-0150563-05
£1,041.44/ea
£0.00
£1,041.44/ea £0.00
100 mgQM-0150563-06
100 mgQM-0150563-06
£1,430.24/ea
£0.00
£1,430.24/ea £0.00

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PBRM1-BD2-IN-5 [CAS 2819989-61-0]

PBRM1-BD2-IN-5 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.