PD 136450 [CAS 139067-52-0]

PD 136450 (CAM 1189) is an antagonist for cholecystokinin 2 (CCK2) . PD 136450 exhibits anti-secretory, anxiolytic and anti-ulcer activities, inhibits gastric acid secretion (IC50=1 mg/kg), and ameliorates the haemorrhagic lesions (IC50=4.7 mg/kg) in rats[1].

[139067-52-0]

C35H40N4O6

612.72

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Cholecystokinin Receptor

Room temperature