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PDGFRα kinase-IN-2 [CAS 3066103-58-7]
PDGFRα kinase-IN-2 [CAS 3066103-58-7]
SKU:QM-0013245
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Product Details
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Description
PDGFRα kinase-IN-2 is a potent PDGFR-α inhibitor with an IC50 of 2.1 nM. PDGFRα kinase-IN-2 exhibits anticancer activity against human colon cancer HT-29 cell with an IC50 of 1.48 μM. PDGFRα kinase-IN-2 has anti-angiogenic activity in zebrafish models and low embryonic lethality. PDGFRα kinase-IN-2 can used for the studies of colon cancer and anti-angiogenesis[1].
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CAS Number
[3066103-58-7]
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Molecular Formula
C24H23N5O3
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Molecular Weight
429.47
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Smiles
COC1=CC2=C(NC3=CC=C(NC(NC4=CC=CC(C)=C4)=O)C=C3)N=CN=C2C=C1OC
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Target
PDGFR
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Isoform
PDGFRα
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Shipping Conditions
Room temperature
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PDGFRα kinase-IN-2 [CAS 3066103-58-7]
PDGFRα kinase-IN-2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.