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PDHK-IN-4

PDHK-IN-4

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SKU:QM-0066961-01

£1,154.43 GBP
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  • Description

    PDHK-IN-4 (Compound 30) is a potent inhibitor of PDHK with IC50s of 0.0051 and 0.0122 μM for PDHK2 and PDHK4, repectively. Pyruvate dehydrogenase kinases (PDHKs) are fascinating agent targets for numerous diseases, including diabetes and cancers. PDHK-IN-4 has the potential for the research of cancer diseases[1].

  • Molecular Formula

    C24H25N5O3

  • Molecular Weight

    431.49

  • Smiles

    O=C(C1=CC=C([C@@H]2CN(C3=C4C(NC5=C4C=CC=C5C6CC6)=NC(C)=N3)[C@H](CO)C2)N1)O

  • Target

    PDHK

  • Solubility

    10 mM in DMSO

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

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Variant Variant total Quantity Price Variant total
1 mgQM-0066961-01
1 mgQM-0066961-01
£1,154.43/ea
£0.00
£1,154.43/ea £0.00
5 mgQM-0066961-02
5 mgQM-0066961-02
£2,873.66/ea
£0.00
£2,873.66/ea £0.00
10 mgQM-0066961-03
10 mgQM-0066961-03
£4,744.76/ea
£0.00
£4,744.76/ea £0.00
25 mgQM-0066961-04
25 mgQM-0066961-04
£10,393.30/ea
£0.00
£10,393.30/ea £0.00

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PDHK-IN-4

PDHK-IN-4 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.