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PERK-IN-4-d3
PERK-IN-4-d3
SKU:QM-0146097-01
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Product Details
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Description
PERK-IN-4-d3 is the deuterium labeled PERK-IN-4. PERK-IN-4 is a potent and selective PERK (protein kinase R (PKR) -like endoplasmic reticulum kinase) inhibitor with an IC50 of 0.3 nM. PERK is activated in response to a variety of endoplasmic reticulum stresses implicated in numerous disease states[1].
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Molecular Formula
C24H16D3F4N5O
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Molecular Weight
472.45
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Smiles
NC1=C(C2=NC=N1)C(C3=CC=C4C(CCN4C(CC5=CC(C(F)(F)F)=CC(F)=C5)=O)=C3)=CN2C([2H])([2H])[2H]
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Target
Isotope-Labeled Compounds; PERK
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PERK-IN-4-d3
PERK-IN-4-d3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.