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PF-04802367 [CAS 1962178-27-3]

PF-04802367 [CAS 1962178-27-3]

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QM-0140432-01

£325.81 GBP
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Product Details

  • Description

    PF-04802367 (PF-367) is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay. PF-04802367 shows desirable central nervous system (CNS) properties and potency. PF-04802367 is equally effective at inhibition of the two known GSK-3 isoforms (GSK-3α and GSK-3β) with IC50 values of 10.0 and 9.0 nM in mobility shift assays, respectively[1].

  • CAS Number

    [1962178-27-3]

  • Molecular Formula

    C16H16ClN5O3

  • Molecular Weight

    361.78

  • Smiles

    O=C(C1=C(C2=CC=C(OC)C(Cl)=C2)OC=N1)NCCCN3N=CN=C3

  • Target

    GSK-3

  • Isoform

    GSK-3α; GSK-3β

  • Purity

    98.43

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302

  • Precautions

    H302
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Variant Variant total Quantity Price Variant total
5 mgQM-0140432-01
5 mgQM-0140432-01
£325.81/ea		 £0.00
£325.81/ea £0.00
10 mM - 1 mLQM-0140432-02
10 mM - 1 mLQM-0140432-02
£353.75/ea		 £0.00
£353.75/ea £0.00
10 mgQM-0140432-03
10 mgQM-0140432-03
£464.31/ea		 £0.00
£464.31/ea £0.00
25 mgQM-0140432-04
25 mgQM-0140432-04
£796.01/ea		 £0.00
£796.01/ea £0.00
50 mgQM-0140432-05
50 mgQM-0140432-05
£1,167.80/ea		 £0.00
£1,167.80/ea £0.00
100 mgQM-0140432-06
100 mgQM-0140432-06
£1,614.92/ea		 £0.00
£1,614.92/ea £0.00
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PF-04802367 [CAS 1962178-27-3]

PF-04802367 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.