PITCOIN4

PITCOIN4 is a highly selective Class II Alpha PI3K-C2α inhibitor. PITCOIN4 shows nanomolar inhibition of PI3K-C2α and >100-fold selectivity in a general kinase panel[1].

C30H29N7O3S2

599.73

CC(C)(NC(CC1=CSC(NC(CSC(N2CCC3=CC=CC=C3)=NC4=C(C2=O)N=CC=N4)=O)=N1)=O)C5=CC=CC=C5

PI3K

99.97

DMSO : 125 mg/mL (ultrasonic)

-20°C, 3 years (Powder)

Blue Ice