PKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM. PKA-IN-1 inhibits cAK in a fashion that is competitive with respect to ATP as substrate[1].
CAS Number
[179985-52-5]
Molecular Formula
C13H11N3O
Molecular Weight
225.25
Smiles
CC(NC1=NC(C)=C(C#N)C2=C1C=CC=C2)=O
Target
PKA
Purity
99.82
Solubility
DMSO : 62.5 mg/mL (ultrasonic; warming; heat to 80°C)