PROTAC BRD9-binding moiety 5 [CAS 893633-37-9]

PROTAC BRD9-binding moiety 5 is a selective BRD9 binder with an IC50 value of 4.20 μM, can be used for the synthesis of PROTACs. PROTAC BRD9-binding moiety 5 has antiproliferative activity against cancer cells[1].

[893633-37-9]

C19H18N6O

346.39

CCC1=NN=C2C(NC3=CC(NC(C)=O)=CC=C3)=NC4=C(N12)C=CC=C4

Epigenetic Reader Domain; Ligands for Target Protein for PROTAC

BRD9

10 mM in DMSO

Room temperature